Total Synthesis of (+/-)-Joubertinamine from 3-(3,4-dimethoxyphenyl)-5-bromo-2-pyrone

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초록

The regioselective synthesis and Diels-Alder cycloaddition of 3-(3,4-dimethoxyphenyl)-5-bromo-2-pyrone provided a new efficient synthetic route to joubertinamine (9.6% total yield over 10 steps).

키워드

QUATERNARY CARBON CENTERASYMMETRIC-SYNTHESISSCELETIUM ALKALOIDS(-)-MESEMBRINECYCLOADDITIONJOUBERTINAMINE(+)-MESEMBRINE3,5-DIBROMO-2-PYRONE(+/-)-MESEMBRINECONSTRUCTION
제목
Total Synthesis of (+/-)-Joubertinamine from 3-(3,4-dimethoxyphenyl)-5-bromo-2-pyrone
저자
Tam, Nguyen ThanhCho, Cheon-Gyu
DOI
10.1021/ol071381p
발행일
2007-08
유형
Article
저널명
Organic Letters
9
17
페이지
3391 ~ 3392